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Publications 2006
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List of publications 2006 from the Consortium.
Links to full articles when available. Some journals require subscription.
[ View
abstracts of some of the articles>> ]
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Abadi, A.H., Abou-Seri, S.M., Abdel-Rahman, D.E., Klein, C., Lozach, O. and
Meijer, L.
Synthesis of 3-substituted-2-oxoindole analogues and their evaluation as
kinase inhibitors, anticancer and antiangiogenic agents.
Eur. J. Med. Chem. 2006, 41, 296-305.
Sciencedirect.com>>
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Alakurtti, S., Mäkelä,T., Koskimies, S. and Yli-Kauhaluoma, J.
Pharmacological properties of the ubiquitous natural
product betulin
European Journal of Pharmaceutical Sciences 2006, 29, 1, 1-13.
Sciencedirect.com>> |
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Aloisi A., DI Gregorio S., Stagno F., Guglielmo P., Mannino F., Sormani M.P.,
Bruzzi P., Gambacorti-Passerini C., Saglio G., Venuta S., Giustolisi R.,
Messina A., Vigneri P.G.
BCR-ABL nuclear entrapment kills human CML cells: ex vivo study on 35
patients with the combination of Imatinib Mesylate and Leptomycin B.
Blood, 2006, 107, 1591-98.
Bloodjournal.org >>
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Arrigoni G., Resjo S., Levander F., Nilsson R., Degerman E., Quadroni M.,
Pinna L. A., and James P. (2006)
Chemical derivatization of phosphoserine and phosphothreonine containing
peptides to increase sensitivity for MALDI-based analysis and for
selectivity of MS/MS analysis
Proteomics 6, 757-766.
http://www3.interscience.wiley.com |
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Assouline S., Laneuville P., Gambacorti-Passerini C.
Panniculitis during Dasatinib Therapy for Imatinib-Resistant Chronic
Myelogenous Leukemia.
New Engl. J of Med, 2006, 354, 2623-2625.
http://content.nejm.org/>>
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Barluenga, S., Dakas, P.Y., Ferandin, Y.,
Meijer, L. and Winssinger, N.
Modular asymmetric synthesis of Aigialomycin D, a kinase-inhibitory
scaffold.
Angew. Chem. Ind. Ed. Engl. 2006, 45, 3951-354.
http://www3.interscience.wiley.com >>
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Bustos V. H., Ferrarese A., Venerando A., Marin O., Allende J. E., and Pinna
L. A. (2006)
The
first armadillo repeat is involved in the recognition and regulation of
beta-catenin phosphorylation by protein kinase CK1.
Proc. Natl. Acad. Sci. U S A. 103, 19725-19730.
http://www.pnas.org
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Coluccia A.M.L., Benati D., Dekhil H., Lan C., Marchesi E.,
Gambacorti-Passerini C.
Inhibition of Src-mediated beta-Catenin tyrosine phosphorylation in
Colorectal cancer cells leads to decreased transcriptional activity and
induces a proliferation block.
Cancer Res., 2006, 66, 2279-86.
http://cancerres.aacrjournals.org >>
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Cozza G., Bonvini P., Zorzi E.,
Poletto G., Pagano M. A., Sarno S., Donella-Deana A., Zagotto G., Rosolen
A., Pinna L. A., Meggio F., and Moro S. (2006)
Identification
of ellagic acid as potent inhibitor of protein kinase CK2: a successful
example of a virtual screening application.
J Med. Chem. 49, 2363-2366.
http://pubs.acs.org
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Gambacorti-Passerini C.
Prognostic variables in patients with chronic myeloid leukemia treated
with imatinib.
Haematologica. 2006, 91, 145.
www.haematologica.org >> |
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Kunick C., Bleeker C. Pruehs C., Totzke F.,
Schaechtele C., Kubbutat M. H. G. and Link A.
Matrix COMPARE analysis discriminates subtle structural differences in a
family of novel antiproliferative agents,
diaryl-3-hydroxy-2,3,3a,10a-tetrahydro-benzo[b]cylopenta[e]
azepine-4,10(1H,5H)-diones.
Bioorg. Med. Chem. Lett. 2006, 16, 2148-2153.
Sciencedirect.com >>
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Kunick, C., Lemcke, T., Meijer, L.:
Paullones
In: Inhibitors of cyclin-dependent kinases as antitumor agents, P. J. Smith,
E. Yue (Editors), CRC Press LLC, Boca Raton (USA), 2006, 227-249. |
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Meijer, L., Guyard, N., Skaltsounis, L.A. and Eisenbrand, G. (Editors) 2006.
“Indirubin, the red shade of indigo”. Editions
« Life in Progress
», Station Biologique, Roscoff, (27 chapters), 297 pp.
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Pagano M. A., Cesaro L., Meggio F., Pinna L. A. (2006)
Protein kinase CK2: a newcomer in the 'druggable kinome'.
Biochem. Soc. Trans. 34, 1303-1306.
[ PDF ]
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Ribas, J., Boix, J. and Meijer, L.
(R)-Roscovitine (CYC202, Seliciclib) sensitizes SH-SY5Y neuroblastoma
cells to Nutlin-3 induced apoptosis.
Exp. Cell Res. 2006, 312, 12, 2394-2400.
Sciencedirect.com>>
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Ribas, J., Bettayeb, K., Ferandin, Y., Knockaert, M., Totzke, F., Schächtele,
C., Mester, J., Polychronopoulos, P., Magiatis, P., Skaltsounis, A.L., Boix,
J. and Meijer, L.
7-bromoindirubin-3’-oxime induces caspase-independent cell death.
Oncogene, 2006.
www.nature.com >>
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Routier, S., Mérour, J.Y.,
Dias, N., Lansiaux, A., Bailly, C., Lozach, O. and Meijer, L..
Synthesis and biological evaluation of novel phenylcarbazoles as potential
anticancer agents.
J. Med. Chem. 2006, 49, 789-799.
Abstract >>
Full article available at:
http://pubs.acs.org
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Ruzza P., Cesaro L., Tourwe D., Calderan A., Biondi B., Maes V., Menegazzo
I., Osler A., Rubini C., Guiotto A., Pinna L. A., Borin G., and Donella-Deana
A. (2006)
Spatial
conformation and topography of the tyrosine aromatic ring in substrate
recognition by protein tyrosine kinases
J Med. Chem. 49, 1916-1924.
http://pubs.acs.org
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Ruzza P., Siligardi G., Donella-Deana A., Calderan A., Hussain R., Rubini
C., Cesaro L., Osler A., Guiotto A., Pinna L. A., and Borin G. (2006)
4-Fluoroproline derivative peptides: effect on PPII conformation and SH3
affinity
J. Pept. Sci. 12, 462-471.
http://www3.interscience.wiley.com>>
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Salvi M., Sarno S., Marin O., Meggio F., Itarte E. and Pinna L. A. (2006)
Discrimination between the activity of protein kinase CK2 holoenzyme and its
catalytic subunits
FEBS Lett. 580, 3948-3952.
Sciencedirect.com>> |
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Testard, A., Logé, C., Léger, B., Robert, J.M., Lozach, O., Blairvacq, M.,
Meijer, L., Thiéry, V. and Besson, T.
Thiazolo[5,4-f]quinazolin-9-one derivatives, inhibitors of glycogen
synthase kinase-3ß.
Bioorg. Med. Chem. Lett. 2006, 16, 3419-3423.
Sciencedirect.com>>
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Tibaldi E., Arrigoni G., Brunati A. M., James P., and Pinna L. A. (2006)
Analysis of a sub-proteome which co-purifies with and is phosphorylated by
the Golgi casein kinase
Cell Mol. Life Sci. 63, 378-389.
http://www.springerlink.com>> |
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Trapp, J., Jochum, A., Meier, R., Saunders, L., Marshall, B., Kunick, C.,
Verdin, E., Goekjian, P., Sippl, W., Jung, M.:
Adenosine mimetics as inhibitors of NAD+-dependent histone deacetylases -
from kinase to sirtuin inhibition
J. Med. Chem. 2006, 49, 7307-7316.
ACS
Publications >>
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Vandromme, L., Piguel, S., Lozach, O., Meijer, L., Legraverend, M., and
Grierson, D.S.
Suzuki-type Pd(0) coupling reactions in the synthesis of 2-arylpurines as
CDK inhibitors.
Bioorg. Med. Chem. Lett. 2006, 16, 3144-3146.
Sciencedirect.com>>
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Updated 24 July 2008
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